| Synthesis of 4-benzyl-1, 3-thiazole derivatives as potential anti-inflammatory agents: an analogue-based drug design approach RN Sharma, FP Xavier, KK Vasu, SC Chaturvedi, SS Pancholi Journal of enzyme inhibition and medicinal chemistry 24 (3), 890-897, 2009 | 261 | 2009 |
| Design, synthesis and characterization of novel 2-(2, 4-disubstituted-thiazole-5-yl)-3-aryl-3H-quinazoline-4-one derivatives as inhibitors of NF-κB and AP-1 mediated … RS Giri, HM Thaker, T Giordano, J Williams, D Rogers, V Sudersanam, ... European journal of medicinal chemistry 44 (5), 2184-2189, 2009 | 230 | 2009 |
| Novel drug designing approach for dual inhibitors as anti-inflammatory agents: implication of pyridine template AD Pillai, PD Rathod, PX Franklin, M Patel, M Nivsarkar, KK Vasu, H Padh, ... Biochemical and Biophysical Research Communications 301 (1), 183-186, 2003 | 130 | 2003 |
| 2-Amino-5-thiazolyl motif: A novel scaffold for designing anti-inflammatory agents of diverse structures PX Franklin, AD Pillai, PD Rathod, S Yerande, M Nivsarkar, H Padh, ... European journal of medicinal chemistry 43 (1), 129-134, 2008 | 124 | 2008 |
| Syntheses of new tetrasubstituted thiophenes as novel anti-inflammatory agents KI Molvi, KK Vasu, SG Yerande, V Sudarsanam, N Haque European journal of medicinal chemistry 42 (8), 1049-1058, 2007 | 96 | 2007 |
| Investigation of microemulsion system for transdermal delivery of itraconazole A Chudasama, V Patel, M Nivsarkar, K Vasu, C Shishoo Journal of advanced pharmaceutical technology & research 2 (1), 30-38, 2011 | 89 | 2011 |
| Tetra substituted thiophenes as anti-inflammatory agents: exploitation of analogue-based drug design AD Pillai, PD Rathod, FP Xavier, H Padh, V Sudarsanam, KK Vasu Bioorganic & medicinal chemistry 13 (24), 6685-6692, 2005 | 87 | 2005 |
| QSAR studies on some thiophene analogs as anti-inflammatory agents: enhancement of activity by electronic parameters and its utilization for chemical lead optimization AD Pillai, S Rani, PD Rathod, FP Xavier, KK Vasu, H Padh, ... Bioorganic & medicinal chemistry 13 (4), 1275-1283, 2005 | 74 | 2005 |
| Design, synthesis and evaluation of novel 2-thiophen-5-yl-3H-quinazolin-4-one analogues as inhibitors of transcription factors NF-кB and AP-1 mediated transcriptional … RS Giri, HM Thaker, T Giordano, J Williams, D Rogers, KK Vasu, ... Bioorganic & Medicinal Chemistry 18 (7), 2796-2808, 2010 | 63 | 2010 |
| Dissolution test for site-specific release isoniazid pellets in USP apparatus 3 (reciprocating cylinder): optimization using response surface methodology A Joshi, S Pund, M Nivsarkar, K Vasu, C Shishoo European journal of pharmaceutics and biopharmaceutics 69 (2), 769-775, 2008 | 63 | 2008 |
| Gastroretentive delivery of rifampicin: In vitro mucoadhesion and in vivo gamma scintigraphy S Pund, A Joshi, K Vasu, M Nivsarkar, C Shishoo International journal of pharmaceutics 411 (1-2), 106-112, 2011 | 59 | 2011 |
| Design, synthesis, and pharmacological evaluation of some 2-[4-morpholino]-3-aryl-5-substituted thiophenes as novel anti-inflammatory agents: generation of a novel anti … AD Pillai, PD Rathod, FP Xavier, KK Vasu, H Padh, V Sudarsanam Bioorganic & medicinal chemistry 12 (17), 4667-4671, 2004 | 56 | 2004 |
| Design, synthesis, and SAR studies of some 5-aliphatic oximino esters of thiophene as potential anti-inflammatory leads: comparative biological activity profile of aliphatic … AD Pillai, PD Rathod, PX Franklin, H Padh, KK Vasu, V Sudarsanam Biochemical and biophysical research communications 317 (4), 1067-1074, 2004 | 47 | 2004 |
| Synthesis and evaluation of quinazolinone derivatives as inhibitors of NF-κB, AP-1 mediated transcription and eIF-4E mediated translational activation: Inhibitors of multi … RS Giri, HM Thaker, T Giordano, B Chen, S Nuthalapaty, KK Vasu, ... European journal of medicinal chemistry 45 (9), 3558-3563, 2010 | 44 | 2010 |
| 2-Amino-5-benzoyl-4-phenylthiazoles: Development of potent and selective adenosine A1 receptor antagonists AB Scheiff, SG Yerande, A El-Tayeb, W Li, GS Inamdar, KK Vasu, ... Bioorganic & Medicinal Chemistry 18 (6), 2195-2203, 2010 | 39 | 2010 |
| Design, synthesis and biological evaluation of novel pyrazolo-pyrimidinones as DPP-IV inhibitors in diabetes SR Sagar, JK Agarwal, DH Pandya, RP Dash, M Nivsarkar, KK Vasu Bioorganic & Medicinal Chemistry Letters 25 (20), 4428-4433, 2015 | 36 | 2015 |
| Multivariate optimization of formulation and process variables influencing physico-mechanical characteristics of site-specific release isoniazid pellets S Pund, A Joshi, K Vasu, M Nivsarkar, C Shishoo International journal of pharmaceutics 388 (1-2), 64-72, 2010 | 36 | 2010 |
| New insight into adenosine receptors selectivity derived from a novel series of [5-substituted-4-phenyl-1, 3-thiazol-2-yl] benzamides and furamides GS Inamdar, AN Pandya, HM Thakar, V Sudarsanam, S Kachler, ... European Journal of Medicinal Chemistry 63, 924-934, 2013 | 33 | 2013 |
| Cyclization of active methylene isocyanides with α-oxodithioesters induced by base: An expedient synthesis of 4-methylthio/ethoxycarbonyl-5-acylthiazoles KR Kiran, TR Swaroop, N Rajeev, SM Anil, KS Rangappa, MP Sadashiva Synthesis 52 (09), 1444-1450, 2020 | 31 | 2020 |
| A convenient synthesis of di-and trisubstituted 2-aminoimidazoles from 1-amidino-3-trityl-thioureas JC Kaila, AB Baraiya, AN Pandya, HB Jalani, KK Vasu, V Sudarsanam Tetrahedron Letters 50 (27), 3955-3958, 2009 | 30 | 2009 |
Amit PandyaMilliporeSigmaVerified email at milliporesigma.com
