| Low intrinsic efficacy for G protein activation can explain the improved side effect profiles of new opioid agonists A Gillis, AB Gondin, A Kliewer, J Sanchez, HD Lim, C Alamein, ... Science signaling 13 (625), eaaz3140, 2020 | 244 | 2020 |
| An overview of late-stage functionalization in today’s drug discovery M Moir, JJ Danon, TA Reekie, M Kassiou Expert opinion on drug discovery 14 (11), 1137-1149, 2019 | 168 | 2019 |
| Cubanes in medicinal chemistry TA Reekie, CM Williams, LM Rendina, M Kassiou Journal of medicinal chemistry 62 (3), 1078-1095, 2018 | 117 | 2018 |
| Body temperature and cardiac changes induced by peripherally administered oxytocin, vasopressin and the non‐peptide oxytocin receptor agonist WAY 267,464: a biotelemetry study … C Hicks, L Ramos, T Reekie, GH Misagh, R Narlawar, M Kassiou, ... British journal of pharmacology 171 (11), 2868-2887, 2014 | 86 | 2014 |
| Comparative evaluation of three TSPO PET radiotracers in a LPS-induced model of mild neuroinflammation in rats S Sridharan, FX Lepelletier, W Trigg, S Banister, T Reekie, M Kassiou, ... Molecular Imaging and Biology 19, 77-89, 2017 | 78 | 2017 |
| The evolving science of phytocannabinoids TA Reekie, MP Scott, M Kassiou Nature Reviews Chemistry 2 (1), 0101, 2017 | 75 | 2017 |
| Peptides, peptidomimetics, and carbohydrate–peptide conjugates as amyloidogenic aggregation inhibitors for Alzheimer’s disease P Ryan, B Patel, V Makwana, HR Jadhav, M Kiefel, A Davey, TA Reekie, ... ACS chemical neuroscience 9 (7), 1530-1551, 2018 | 73 | 2018 |
| Imaging glial activation in patients with post-treatment Lyme disease symptoms: a pilot study using [11C]DPA-713 PET JM Coughlin, T Yang, AW Rebman, KT Bechtold, Y Du, WB Mathews, ... Journal of Neuroinflammation 15, 1-7, 2018 | 63 | 2018 |
| Application of a Raney-Cobalt-Mediated Tandem Reductive Cyclization Protocol to Total Syntheses of the Aspidosperma Alkaloids (±)-Limaspermidine and (±)-1 … SH Tan, MG Banwell, AC Willis, TA Reekie Organic letters 14 (22), 5621-5623, 2012 | 61 | 2012 |
| Challenges and opportunities in central nervous system drug discovery JJ Danon, TA Reekie, M Kassiou Trends in Chemistry 1 (6), 612-624, 2019 | 54 | 2019 |
| Targeting the oxytocin system: new pharmacotherapeutic approaches D Gulliver, E Werry, TA Reekie, TA Katte, W Jorgensen, M Kassiou Trends in pharmacological sciences 40 (1), 22-37, 2019 | 54 | 2019 |
| In vivo assessment of neuroinflammation in progressive multiple sclerosis: a proof of concept study with [18F]DPA714 PET MHJ Hagens, SV Golla, MT Wijburg, M Yaqub, D Heijtel, MD Steenwijk, ... Journal of neuroinflammation 15, 1-10, 2018 | 54 | 2018 |
| Prodromal neuroinflammatory, cholinergic and metabolite dysfunction detected by PET and MRS in the TgF344-AD transgenic rat model of AD: a collaborative multi-modal study AM Chaney, FR Lopez-Picon, S Serrière, R Wang, D Bochicchio, ... Theranostics 11 (14), 6644, 2021 | 47 | 2021 |
| Structural optimization and pharmacological evaluation of inhibitors targeting dual-specificity tyrosine phosphorylation-regulated kinases (DYRK) and CDC-like kinases (CLK) in … Q Zhou, AF Phoa, RH Abbassi, M Hoque, TA Reekie, JS Font, RM Ryan, ... Journal of Medicinal Chemistry 60 (5), 2052-2070, 2017 | 46 | 2017 |
| Synthesis of biologically active seven-membered-ring heterocycles TA Reekie, ME Kavanagh, M Longworth, M Kassiou Synthesis, 3211-3227, 2013 | 40 | 2013 |
| A Raney-Cobalt-Mediated Tandem Reductive Cyclization Route to the 1,5-Methanoazocino[4,3-b]indole Framework of the Uleine and Strychnos Alkaloids TA Reekie, MG Banwell, AC Willis The Journal of Organic Chemistry 77 (23), 10773-10781, 2012 | 38 | 2012 |
| The chemoenzymatic total synthesis of phellodonic acid, a biologically active and highly functionalized hirsutane derivative isolated from the tasmanian fungus Phellodon melaleucus TA Reekie, KAB Austin, MG Banwell, AC Willis Australian Journal of Chemistry 61 (2), 94-106, 2008 | 35 | 2008 |
| Synthesis of usnic acid derivatives and evaluation of their antiproliferative activity against cancer cells A Pyrczak-Felczykowska, R Narlawar, A Pawlik, B Guzow-Krzemińska, ... Journal of natural products 82 (7), 1768-1778, 2019 | 33 | 2019 |
| RANEY® cobalt–an underutilised reagent for the selective cleavage of C–X and N–O bonds MG Banwell, MT Jones, TA Reekie, BD Schwartz, SH Tan, LV White Organic & biomolecular chemistry 12 (38), 7433-7444, 2014 | 33 | 2014 |
| Chemoenzymatic methods for the enantioselective assembly of bioactive natural products KAB Austin, M Matveenko, TA Reekie, MG Banwell Chemistry in Australia 75 (11), 2008 | 31 | 2008 |
Michael KassiouProfessor of Medicinal Chemistry, The University of SydneyVerified email at sydney.edu.au
