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Arthur Christopoulos
Arthur Christopoulos
Verified email at monash.edu - Homepage
Title
Cited by
Cited by
Year
Fitting models to biological data using linear and nonlinear regression: a practical guide to curve fitting
AC Harvey Motulsky
Oxford University Press, 2004
35002004
Strategies to address low drug solubility in discovery and development
HD Williams, NL Trevaskis, SA Charman, RM Shanker, WN Charman, ...
Pharmacological reviews 65 (1), 315-499, 2013
17822013
Functional selectivity and classical concepts of quantitative pharmacology
JD Urban, WP Clarke, M Von Zastrow, DE Nichols, B Kobilka, H Weinstein, ...
Journal of Pharmacology and Experimental Therapeutics 320 (1), 1-13, 2007
13392007
Allosteric modulators of GPCRs: a novel approach for the treatment of CNS disorders
P Jeffrey Conn, A Christopoulos, CW Lindsley
Nature reviews Drug discovery 8 (1), 41-54, 2009
12252009
G protein-coupled receptor allosterism and complexing
A Christopoulos, T Kenakin
Pharmacological reviews 54 (2), 323-374, 2002
10422002
Activation and allosteric modulation of a muscarinic acetylcholine receptor
AC Kruse, AM Ring, A Manglik, J Hu, K Hu, K Eitel, H Hübner, E Pardon, ...
Nature 504 (7478), 101-106, 2013
10042013
International Union of Pharmacology Committee on Receptor Nomenclature and Drug Classification. XXXVIII. Update on terms and symbols in quantitative pharmacology
RR Neubig, M Spedding, T Kenakin, A Christopoulos
Pharmacological reviews 55 (4), 597-606, 2003
8472003
Allosteric binding sites on cell-surface receptors: novel targets for drug discovery
A Christopoulos
Nature reviews Drug discovery 1 (3), 198-210, 2002
8412002
Signalling bias in new drug discovery: detection, quantification and therapeutic impact
T Kenakin, A Christopoulos
Nature reviews Drug discovery 12 (3), 205-216, 2013
8332013
Allosteric modulation of G protein–coupled receptors
LT May, K Leach, PM Sexton, A Christopoulos
Annu. Rev. Pharmacol. Toxicol. 47 (1), 1-51, 2007
8322007
The Concise Guide to PHARMACOLOGY 2019/20: G protein‐coupled receptors
SPH Alexander, A Christopoulos, AP Davenport, E Kelly, A Mathie, ...
British journal of pharmacology 176, S21-S141, 2019
8032019
Mechanisms of signalling and biased agonism in G protein-coupled receptors
D Wootten, A Christopoulos, M Marti-Solano, MM Babu, PM Sexton
Nature reviews Molecular cell biology 19 (10), 638-653, 2018
6822018
The Concise Guide to PHARMACOLOGY 2017/18: G protein‐coupled receptors
SPH Alexander, A Christopoulos, AP Davenport, E Kelly, NV Marrion, ...
British journal of pharmacology 174, S17-S129, 2017
6812017
G-protein–coupled receptor Mas is a physiological antagonist of the angiotensin II type 1 receptor
E Kostenis, G Milligan, A Christopoulos, CF Sanchez-Ferrer, ...
Circulation 111 (14), 1806-1813, 2005
5532005
Emerging paradigms in GPCR allostery: implications for drug discovery
D Wootten, A Christopoulos, PM Sexton
Nature reviews Drug discovery 12 (8), 630-644, 2013
5462013
Allosteric modulation of the cannabinoid CB1 receptor
MR Price, GL Baillie, A Thomas, LA Stevenson, M Easson, R Goodwin, ...
Molecular pharmacology 68 (5), 1484-1495, 2005
5122005
Phase-plate cryo-EM structure of a class B GPCR–G-protein complex
YL Liang, M Khoshouei, M Radjainia, Y Zhang, A Glukhova, J Tarrasch, ...
Nature 546 (7656), 118-123, 2017
5112017
A simple method for quantifying functional selectivity and agonist bias
T Kenakin, C Watson, V Muniz-Medina, A Christopoulos, S Novick
ACS chemical neuroscience 3 (3), 193-203, 2012
5082012
The Concise Guide to PHARMACOLOGY 2021/22: G protein‐coupled receptors
SPH Alexander, A Christopoulos, AP Davenport, E Kelly, A Mathie, ...
British journal of pharmacology 178, S27-S156, 2021
5032021
Muscarinic acetylcholine receptors: novel opportunities for drug development
AC Kruse, BK Kobilka, D Gautam, PM Sexton, A Christopoulos, J Wess
Nature reviews Drug discovery 13 (7), 549-560, 2014
4742014
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