Intramolecular Friedel–Crafts acylation reaction promoted by 1, 1, 1, 3, 3, 3-hexafluoro-2-propanol HF Motiwala, RH Vekariya, J Aube Organic letters 17 (21), 5484-5487, 2015 | 154 | 2015 |
Mephedrone and methylenedioxypyrovalerone (MDPV), major constituents of “bath salts,” produce opposite effects at the human dopamine transporter K Cameron, R Kolanos, R Verkariya, L De Felice, RA Glennon Psychopharmacology 227, 493-499, 2013 | 129 | 2013 |
Hexafluoro-2-propanol-promoted intermolecular Friedel–Crafts acylation reaction RH Vekariya, J Aube Organic letters 18 (15), 3534-3537, 2016 | 121 | 2016 |
A concomitant allylic azide rearrangement/intramolecular azide–alkyne cycloaddition sequence RH Vekariya, R Liu, J Aubé Organic letters 16 (7), 1844-1847, 2014 | 55 | 2014 |
A novel mu-delta opioid agonist demonstrates enhanced efficacy with reduced tolerance and dependence in mouse neuropathic pain models W Lei, RH Vekariya, S Ananthan, JM Streicher The journal of pain 21 (1-2), 146-160, 2020 | 41 | 2020 |
Abuse-related neurochemical and behavioral effects of cathinone and 4-methylcathinone stereoisomers in rats BA Hutsell, MH Baumann, JS Partilla, ML Banks, R Vekariya, RA Glennon, ... European Neuropsychopharmacology 26 (2), 288-297, 2016 | 26 | 2016 |
Synthesis and structure–activity relationships of 5′-aryl-14-alkoxypyridomorphinans: Identification of a μ opioid receptor agonist/δ opioid receptor antagonist ligand with … RH Vekariya, W Lei, A Ray, SK Saini, S Zhang, G Molnar, D Barlow, ... Journal of medicinal chemistry 63 (14), 7663-7694, 2020 | 24 | 2020 |
Targeting the HuR oncogenic role with a new class of cytoplasmic dimerization inhibitors N Filippova, X Yang, S Ananthan, J Calano, V Pathak, L Bratton, ... Cancer research 81 (8), 2220-2233, 2021 | 22 | 2021 |
Structure-Activity Investigation of a G Protein-Biased Agonist Reveals Molecular Determinants for Biased Signaling of the D2 Dopamine Receptor LS Chun, RH Vekariya, RB Free, Y Li, DT Lin, P Su, F Liu, Y Namkung, ... Frontiers in synaptic neuroscience 10, 2, 2018 | 17 | 2018 |
Reformulating a Pharmacophore for 5-HT2A Serotonin Receptor Antagonists J Younkin, SA Gaitonde, A Ellaithy, R Vekariya, L Baki, JL Moreno, ... ACS chemical neuroscience 7 (9), 1292-1299, 2016 | 13 | 2016 |
One-Pot Synthesis of [1, 2, 3] Triazolo [1, 5-a] quinoxalin-4 (5H)-ones by a Metal-Free Sequential Ugi-4CR/Alkyne–Azide Cycloaddition Reaction YM Yan, HY Li, M Zhang, RX Wang, CG Zhou, ZX Ren, MW Ding Synlett 31 (01), 73-76, 2020 | 11 | 2020 |
SRI-32743, a novel allosteric modulator, attenuates HIV-1 Tat protein-induced inhibition of the dopamine transporter and alleviates the potentiation of cocaine reward in HIV-1 … J Zhu, PM Quizon, Y Wang, CA Adeniran, MJ Strauss, AC Jiménez-Torres, ... Neuropharmacology 220, 109239, 2022 | 9 | 2022 |
Direct Deoxygenative Intramolecular Acylation of Biarylcarboxylic Acids Y Li, W Xu, C Zhu, J Xie Synlett 32 (04), 387-390, 2021 | 5 | 2021 |
Towards understanding the mechanism of action of abused cathinones R Vekariya | 2 | 2012 |
Hexafluoro‐2‐propanol‐promoted Intramolecular Friedel‐Crafts Acylation RH Vekariya, MC Horton, J Aubé* Organic Syntheses 95, 486-499, 2018 | 1 | 2018 |
ORIC-613, a potential first-and best-in-class, orally bioavailable, potent and selective PLK4 inhibitor with synthetic lethality in TRIM37 high cancer models KA Edgar, S McRee, G Andretta, C Chen, C Colas, W Fang, W Kong, ... Cancer Research 84 (6_Supplement), 594-594, 2024 | | 2024 |
Selective PLK4 Inhibitors Demonstrate Synthetic Lethality in TRIM37 Amplified Neuroblastoma and Breast Cancer Models While Less Selective Inhibitors Do Not SK McRee, X Chen, C Colas, A Daemen, W Fang, W Kong, J Long, F Liu, ... | | 2023 |
Not Logged In Login JJ Topczewski, MR Porter Synlett 29 (12), 1537-1542, 2018 | | 2018 |
Studies and Synthetic Methodology: 1. Cycloaddition of Allylic Azides and Alkynes, 2. Hexafluoro-2-propanol-promoted Friedel–Crafts Acylation Reactions RH Vekariya University of Kansas, 2016 | | 2016 |
Friedel-Crafts chemistry in HFIP R Vekariya, H Motiwala, S Roy, M Bovino, J Aube ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 252, 2016 | | 2016 |