Constraining cyclic peptides to mimic protein structure motifs TA Hill, NE Shepherd, F Diness, DP Fairlie Angewandte Chemie International Edition 53 (48), 13020-13041, 2014 | 424 | 2014 |
Comparative α‐Helicity of cyclic pentapeptides in water AD De Araujo, HN Hoang, WM Kok, F Diness, P Gupta, TA Hill, RW Driver, ... Angewandte Chemie International Edition 53 (27), 6965-6969, 2014 | 187 | 2014 |
Recent fascinating aspects of the CuAAC click reaction M Meldal, F Diness Trends in Chemistry 2 (6), 569-584, 2020 | 168 | 2020 |
Catalyst‐Free N‐Arylation Using Unactivated Fluorobenzenes F Diness, DP Fairlie Angewandte Chemie International Edition 32 (51), 8012-8016, 2012 | 135 | 2012 |
Rational tuning of fluorobenzene probes for Cysteine‐Selective protein modification AM Embaby, S Schoffelen, C Kofoed, M Meldal, F Diness Angewandte Chemie 130 (27), 8154-8158, 2018 | 71 | 2018 |
The Pictet-Spengler reaction in solid-phase combinatorial chemistry. TE Nielsen, F Diness, M Meldal Current Opinion in Drug Discovery & Development 6 (6), 801-814, 2003 | 71 | 2003 |
Total synthesis, structure, and oral absorption of a thiazole cyclic peptide, sanguinamide A DS Nielsen, HN Hoang, RJ Lohman, F Diness, DP Fairlie Organic letters 14 (22), 5720-5723, 2012 | 69 | 2012 |
Fixierung cyclischer Peptide: Mimetika von Proteinstrukturmotiven TA Hill, NE Shepherd, F Diness, DP Fairlie Angewandte Chemie 126 (48), 13234-13257, 2014 | 58 | 2014 |
Mechanism and Scope of Base‐Controlled Catalyst‐Free N‐Arylation of Amines with Unactivated Fluorobenzenes C Borch Jacobsen, M Meldal, F Diness Chemistry–A European Journal 23 (4), 846-851, 2017 | 46 | 2017 |
Solid‐Phase Synthesis of Tetrahydro‐β‐carbolines and Tetrahydroisoquinolines by Stereoselective Intramolecular N‐Carbamyliminium Pictet–Spengler Reactions F Diness, J Beyer, M Meldal Chemistry–A European Journal 12 (31), 8056-8066, 2006 | 43 | 2006 |
Probing the aglycon binding site of a β-glucosidase: a collection of C-1-modified 2, 5-dideoxy-2, 5-imino-d-mannitol derivatives and their structure–activity relationships as … TM Wrodnigg, F Diness, C Gruber, H Häusler, I Lundt, K Rupitz, ... Bioorganic & medicinal chemistry 12 (13), 3485-3495, 2004 | 41 | 2004 |
Sequential Direct SNAr Reactions of Pentafluorobenzenes with Azole or Indole Derivatives F Diness, M Begtrup Organic letters 16 (11), 3130-3133, 2014 | 39 | 2014 |
C-Terminally modified peptides via cleavage of the HMBA linker by O-, N-or S-nucleophiles J Hansen, F Diness, M Meldal Organic & Biomolecular Chemistry 14 (12), 3238-3245, 2016 | 35 | 2016 |
Synthesis of 3‐Boc‐(1, 3)‐oxazinane‐Protected Amino Aldehydes from Amino Acids and Their Conversion into Urea Precursors. Novel Building Blocks for Combinatorial Synthesis F Diness, J Beyer, M Meldal QSAR & Combinatorial Science 23 (2‐3), 130-144, 2004 | 27 | 2004 |
Synthesis of the thiazole–thiazoline fragment of largazole analogues F Diness, DS Nielsen, DP Fairlie The Journal of Organic Chemistry 76 (23), 9845-9851, 2011 | 26 | 2011 |
Click-chemistry-mediated synthesis of selective melanocortin receptor 4 agonists D Palmer, JPL Gonçalves, L V. Hansen, B Wu, H Hald, S Schoffelen, ... Journal of Medicinal Chemistry 60 (21), 8716-8730, 2017 | 21 | 2017 |
Biophysical characterization of the proton-coupled oligopeptide transporter YjdL JM Jensen, FC Simonsen, A Mastali, H Hald, I Lillebro, F Diness, L Olsen, ... Peptides 38 (1), 89-93, 2012 | 19 | 2012 |
Ralph F. Hirschmann award address 2009: Merger of organic chemistry with peptide diversity M Meldal, CW Tornøe, TE Nielsen, F Diness, ST Le Quement, ... Peptide Science: Original Research on Biomolecules 94 (2), 161-182, 2010 | 19 | 2010 |
Chemical modification of proteins–challenges and trends at the start of the 2020s NH Fischer, MT Oliveira, F Diness Biomaterials Science 11 (3), 719-748, 2023 | 16 | 2023 |
Imidazolones in Diastereoselective Cyclization Reactions and CuII‐Catalysed Cross‐Coupling Reactions F Diness, M Meldal Chemistry–A European Journal 15 (29), 7044-7047, 2009 | 15 | 2009 |