| Acylhydrazone derivatives: a patent review RC Maia, R Tesch, CAM Fraga Expert opinion on therapeutic patents 24 (11), 1161-1170, 2014 | 65 | 2014 |
| Antihypertensive profile of 2-thienyl-3, 4-methylenedioxybenzoylhydrazone is mediated by activation of the A2A adenosine receptor CM Leal, SL Pereira, AE Kümmerle, DM Leal, R Tesch, ... European journal of medicinal chemistry 55, 49-57, 2012 | 50 | 2012 |
| N-acylhydrazone derivative ameliorates monocrotaline-induced pulmonary hypertension through the modulation of adenosine AA2R activity AKN Alencar, SL Pereira, FE da Silva, LVP Mendes, V do MN Cunha, ... International journal of cardiology 173 (2), 154-162, 2014 | 44 | 2014 |
| Phenylpiperazine derivatives: a patent review (2006–present) RC Maia, R Tesch, CAM Fraga Expert opinion on therapeutic patents 22 (10), 1169-1178, 2012 | 29 | 2012 |
| Structure-based design of selective salt-inducible kinase inhibitors R Tesch, M Rak, M Raab, LM Berger, T Kronenberger, AC Joerger, ... Journal of Medicinal Chemistry 64 (12), 8142-8160, 2021 | 28 | 2021 |
| Pyridinylimidazoles as dual glycogen synthase kinase 3β/p38α mitogen-activated protein kinase inhibitors F Heider, F Ansideri, R Tesch, T Pantsar, U Haun, E Döring, M Kudolo, ... European journal of medicinal chemistry 175, 309-329, 2019 | 28 | 2019 |
| Fast iterative synthetic approach toward identification of novel highly selective p38 MAP kinase inhibitors S Röhm, BT Berger, M Schröder, A Chaikuad, R Winkel, KFW Hekking, ... Journal of medicinal chemistry 62 (23), 10757-10782, 2019 | 26 | 2019 |
| Novel Potent Imidazo[1,2-a]pyridine-N-Glycinyl-Hydrazone Inhibitors of TNF-α Production: In Vitro and In Vivo Studies RB Lacerda, NM Sales, LL da Silva, R Tesch, ALP Miranda, EJ Barreiro, ... PLoS One 9 (3), e91660, 2014 | 25 | 2014 |
| The small-molecule inhibitor MRIA9 reveals novel insights into the cell cycle roles of SIK2 in ovarian cancer cells M Raab, M Rak, R Tesch, K Gasimli, S Becker, S Knapp, K Strebhardt, ... Cancers 13 (15), 3658, 2021 | 16 | 2021 |
| A highly selective chemical probe for activin receptor-like kinases ALK4 and ALK5 T Hanke, JF Wong, BT Berger, I Abdi, LM Berger, R Tesch, C Tredup, ... ACS Chemical Biology 15 (4), 862-870, 2020 | 15 | 2020 |
| Addressing a trapped high-energy water: design and synthesis of highly potent pyrimidoindole-based glycogen synthase kinase-3β inhibitors S Andreev, T Pantsar, R Tesch, N Kahlke, A El-Gokha, F Ansideri, ... Journal of Medicinal Chemistry 65 (2), 1283-1301, 2021 | 13 | 2021 |
| An unusual intramolecular halogen bond guides conformational selection R Tesch, C Becker, MP Müller, ME Beck, L Quambusch, M Getlik, ... Angewandte Chemie International Edition 57 (31), 9970-9975, 2018 | 13 | 2018 |
| LASSBio-897 Reduces Lung Injury Induced by Silica Particles in Mice: Potential Interaction with the A2A Receptor VF Carvalho, TPT Ferreira, ACS De Arantes, F Noël, R Tesch, ... Frontiers in Pharmacology 8, 778, 2017 | 7 | 2017 |
| Shifting the selectivity of pyrido [2, 3-d] pyrimidin-7 (8H)-one inhibitors towards the salt-inducible kinase (SIK) subfamily M Rak, R Tesch, LM Berger, E Shevchenko, M Raab, A Tjaden, R Zhubi, ... European Journal of Medicinal Chemistry 254, 115347, 2023 | 5 | 2023 |
| Prevention and Reversal of MorphineInduced Tolerance by Novel Muscarinic Receptor Agonist in Rats with Neuropathic Pain CES Monteiro, N Nascimento-Júnior, M Trachez, R Tesch, T Mendes J Neurol Neurophysiol 6 (282), 2, 2015 | 5 | 2015 |
| The role of natural products on the discovery of new drug candidates for neurogenerative disorders FP Viegas, M RdC, R Tesch Frontiers CNS Drug Discov 2, 2211, 2013 | 2 | 2013 |
| Revisitando o Conceito Mensagem-Endereço em Química Medicinal R Tesch, CMR Sant'Anna, CAM Fraga Revista Virtual de Química 7 (2), 594-608, 2015 | 1 | 2015 |
| Development of Selective Pyrido[2,3-d]pyrimidin-7(8H)-one-Based Mammalian STE20-Like (MST3/4) Kinase Inhibitors M Rak, A Menge, R Tesch, LM Berger, DI Balourdas, E Shevchenko, ... Journal of Medicinal Chemistry 67 (5), 3813-3842, 2024 | | 2024 |
| Refining Selectivity of p38 MAP Kinase Inhibitors D Trauner, M Reynders Synfacts 16 (02), 0219, 2020 | | 2020 |
| Design, Synthesis and Pharmacological Evaluation of Novel Antiinflammatory and Analgesic O-Benzyloxime Compounds Derived From Natural Eugenol R César da Silva, F Veiga, FC Vilela, AV Pereira, ... Letters in Drug Design & Discovery 16 (10), 1157-1166, 2019 | | 2019 |
