Design and Mechanism of (S)-3-Amino-4-(difluoromethylenyl)cyclopent-1-ene-1-carboxylic Acid, a Highly Potent γ-Aminobutyric Acid Aminotransferase Inactivator … JI Juncosa, K Takaya, HV Le, MJ Moschitto, PM Weerawarna, ... Journal of the American Chemical Society 140 (6), 2151-2164, 2018 | 70 | 2018 |
Syntheses of arnottin I and arnottin II MJ Moschitto, DR Anthony, CA Lewis The Journal of organic chemistry 80 (6), 3339-3342, 2015 | 43 | 2015 |
Mechanism of Inactivation of Ornithine Aminotransferase by (1S,3S)-3-Amino-4-(hexafluoropropan-2-ylidenyl)cyclopentane-1-carboxylic Acid MJ Moschitto, PF Doubleday, DS Catlin, NL Kelleher, D Liu, RB Silverman Journal of the American Chemical Society 141 (27), 10711-10721, 2019 | 22 | 2019 |
Synthesis of (S)-3-Amino-4-(difluoromethylenyl)-cyclopent-1-ene-1-carboxylic Acid (OV329), a Potent Inactivator of γ-Aminobutyric Acid Aminotransferase MJ Moschitto, RB Silverman Organic letters 20 (15), 4589-4592, 2018 | 17 | 2018 |
Regiodivergent Addition of Phenols to Allylic Oxides: Control of 1, 2‐and 1, 4‐Additions for Cyclitol Synthesis MJ Moschitto, DN Vaccarello, CA Lewis Angewandte Chemie 127 (7), 2170-2173, 2015 | 12 | 2015 |
Synthesis of Quinoline Silyloxymethylsulfones as Intermediates to Sulfonyl Derivatives TI Patel, R Laha, MJ Moschitto The Journal of Organic Chemistry 87 (22), 15679-15683, 2022 | 7 | 2022 |
Desulfinative Alkylation of Heteroarenes via an Electrostatic Electron Donor–Acceptor Complex R Laha, TI Patel, MJ Moschitto Organic letters 24 (40), 7394-7399, 2022 | 5 | 2022 |
Theoretical and mechanistic validation of global kinetic parameters of the inactivation of GABA aminotransferase by OV329 and CPP-115 PM Weerawarna, MJ Moschitto, RB Silverman ACS chemical biology 16 (4), 615-630, 2021 | 5 | 2021 |
Synthesis of the Rubiyunnanin B Core Aglycon MJ Moschitto, CA Lewis European Journal of Organic Chemistry 2016 (28), 4773-4777, 2016 | 4 | 2016 |
Regiodivergent Addition of Phenols to Allylic Oxides DN Vaccarello, MJ Moschitto, CA Lewis The Journal of organic chemistry 80 (10), 5252-5259, 2015 | 4 | 2015 |
Expanding the 18F-radiochemical space: synthesis and applications of 1, 1-18F-difluorinated alkenes M Tredwell Synlett 30 (12), 1371-1376, 2019 | 3 | 2019 |
Allylic Oxide Regio-Resolution as a Tool for the Synthesis and Transfer of Carbasugars CA Lewis, MJ Moschitto, DN Vaccarello Synlett 26 (18), 2473-2478, 2015 | 1 | 2015 |
Streamlining SuFEx Inhibitor Development: A Unified Approach Using Orthogonal Sulfinate Protecting Groups T Patel, Y Chi, R Laha, M Moschitto | | 2024 |
From TgO/GABA-AT, GABA, and T-263 Mutant to Conception of Toxoplasma J Lykins, MJ Moschitto, Y Zhou, EV Filippova, HV Le, T Tomita, BA Fox, ... Iscience 27 (1), 2024 | | 2024 |
Analogs of 3-amino-4-(propan-2-ylidene) cyclopentane-1-carboxylic acid and uses thereof for treating diseases and disorders associated with ornithine aminotransferase activity RB Silverman, MJ Moschitto US Patent 11,203,596, 2021 | | 2021 |
Process for the synthesis of (s) 3-amino-4-(difluoromethylenyl) cyclopent-1-ene-1-carboxylic acid RB Silverman, M Moschitto US Patent App. 16/950,542, 2021 | | 2021 |
Process for the synthesis of (s) 3-amino-4-(difluoromethylenyl) cyclopent-1-ene-1-carboxylic acid RB Silverman, M Moschitto US Patent 10,836,708, 2020 | | 2020 |
Synthesis of OV329 P Kocienski Synfacts 14 (10), 1011, 2018 | | 2018 |
Synthesis And Manipulation Of Carbasugars And Natural Product Scaffolds M Moschitto | | 2016 |