Microwave assisted synthesis: a new technology in drug discovery V Santagada, F Frecentese, E Perissutti, F Fiorino, B Severino, ... Mini reviews in medicinal chemistry 9 (3), 340-358, 2009 | 135 | 2009 |
5-HT1A Receptor: An Old Target as a New Attractive Tool in Drug Discovery from Central Nervous System to Cancer F Fiorino, B Severino, E Magli, A Ciano, G Caliendo, V Santagada, ... Journal of Medicinal Chemistry 57 (11), 4407-4426, 2014 | 90 | 2014 |
Heavy Metals Size Distribution in PM10 and Environmental-Sanitary Risk Analysis in Acerra (Italy) P Di Vaio, E Magli, G Caliendo, A Corvino, F Fiorino, F Frecentese, ... Atmosphere 9 (2), 58, 2018 | 61 | 2018 |
The Application of Microwaves in Combinatorial and High‐Throughput Synthesis as New Synthetic Procedure in Drug Discovery V Santagada, F Frecentese, E Perissutti, L Favretto, G Caliendo QSAR & Combinatorial Science 23 (10), 919-944, 2004 | 57 | 2004 |
Synthesis and pharmacological evaluations of sildenafil analogues for treatment of erectile dysfunction HA Flores Toque, FBM Priviero, CE Teixeira, E Perissutti, F Fiorino, ... Journal of medicinal chemistry 51 (9), 2807-2815, 2008 | 56 | 2008 |
A suitable 1, 2, 4-oxadiazoles synthesis by microwave irradiation V Santagada, F Frecentese, E Perissutti, D Cirillo, S Terracciano, ... Bioorganic & medicinal chemistry letters 14 (17), 4491-4493, 2004 | 56 | 2004 |
Trends in H2S-Donors Chemistry and Their Effects in Cardiovascular Diseases A Corvino, F Frecentese, E Magli, E Perissutti, V Santagada, ... Antioxidants 10 (3), 429, 2021 | 53 | 2021 |
Level, potential sources of polycyclic aromatic hydrocarbons (PAHs) in particulate matter (PM10) in Naples P Di Vaio, B Cocozziello, A Corvino, F Fiorino, F Frecentese, E Magli, ... Atmospheric environment 129, 186-196, 2016 | 51 | 2016 |
1, 2, 4-Thiadiazolidin-3, 5-diones as novel hydrogen sulfide donors B Severino, A Corvino, F Fiorino, P Luciano, F Frecentese, E Magli, ... European Journal of Medicinal Chemistry 143, 1677-1686, 2018 | 45 | 2018 |
H2S Donors and Their Use in Medicinal Chemistry E Magli, E Perissutti, V Santagada, G Caliendo, A Corvino, G Esposito, ... Biomolecules 11 (12), 1899, 2021 | 37 | 2021 |
Structure-activity relationships study of isothiocyanates for H2S releasing properties: 3-Pyridyl-isothiocyanate as a new promising cardioprotective agent V Citi, A Corvino, F Fiorino, F Frecentese, E Magli, E Perissutti, ... Journal of Advanced Research 27, 41-53, 2021 | 34 | 2021 |
Lipophilic and polar interaction forces between acidic drugs and membrane phospholipids encoded in IAM-HPLC indexes: Their role in membrane partition and relationships with BBB … L Grumetto, C Carpentiero, P Di Vaio, F Frecentese, F Barbato Journal of pharmaceutical and biomedical analysis 75, 165-172, 2013 | 32 | 2013 |
Anti-metastatic properties of naproxen-HBTA in a murine model of cutaneous melanoma G Ercolano, P De Cicco, F Frecentese, I Saccone, A Corvino, F Giordano, ... Frontiers in Pharmacology 10, 66, 2019 | 28 | 2019 |
Synthesis and In‐vitro Pharmacological Evaluation of New 5‐HT1A Receptor Ligands Containing a Benzotriazinone Nucleus F Fiorino, B Severino, F De Angelis, E Perissutti, F Frecentese, ... Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2008 | 28 | 2008 |
The role of 5-HT1A receptor in cancer as a new opportunity in medicinal chemistry A Corvino, F Fiorino, B Severino, I Saccone, F Frecentese, E Perissutti, ... Current Medicinal Chemistry 25 (27), 3214-3227, 2018 | 26 | 2018 |
New 5-HT1A, 5HT2A and 5HT2C receptor ligands containing a picolinic nucleus: Synthesis, in vitro and in vivo pharmacological evaluation F Fiorino, E Magli, E Kędzierska, A Ciano, A Corvino, B Severino, ... Bioorganic & Medicinal Chemistry 25 (20), 5820-5837, 2017 | 26 | 2017 |
Fragment-based de novo design of a cystathionine γ-lyase selective inhibitor blocking hydrogen sulfide production A Corvino, B Severino, F Fiorino, F Frecentese, E Magli, E Perissutti, ... Scientific Reports 6 (1), 34398, 2016 | 26 | 2016 |
Efficient microwave combinatorial parallel and nonparallel synthesis of N-alkylated glycine methyl esters as peptide building blocks V Santagada, F Frecentese, E Perissutti, F Fiorino, B Severino, D Cirillo, ... Journal of Combinatorial Chemistry 7 (4), 618-621, 2005 | 24 | 2005 |
Design, synthesis and biological evaluation of TAR and cTAR binders as HIV-1 nucleocapsid inhibitors A Sosic, F Frecentese, E Perissutti, L Sinigaglia, V Santagada, ... MedChemComm 4 (10), 1388-1393, 2013 | 23 | 2013 |
Kallikrein protease activated receptor (PAR) axis: an attractive target for drug development G Caliendo, V Santagada, E Perissutti, B Severino, F Fiorino, ... Journal of Medicinal Chemistry 55 (15), 6669-6686, 2012 | 20 | 2012 |