| Bafetinib (INNO-406) reverses multidrug resistance by inhibiting the efflux function of ABCB1 and ABCG2 transporters YK Zhang, GN Zhang, YJ Wang, BA Patel, TT Talele, DH Yang, ZS Chen Scientific reports 6 (1), 25694, 2016 | 63 | 2016 |
| Design and synthesis of human ABCB1 (P-glycoprotein) inhibitors by peptide coupling of diverse chemical scaffolds on carboxyl and amino termini of (S)-valine-derived thiazole … S Singh, NR Prasad, EE Chufan, BA Patel, YJ Wang, ZS Chen, ... Journal of Medicinal Chemistry 57 (10), 4058-4072, 2014 | 62 | 2014 |
| Semi-synthetic ocotillol analogues as selective ABCB1-mediated drug resistance reversal agents YK Zhang, H Zhang, GN Zhang, YJ Wang, RJ Kathawala, R Si, BA Patel, ... Oncotarget 6 (27), 24277, 2015 | 43 | 2015 |
| The BTK inhibitor ibrutinib (PCI-32765) overcomes paclitaxel resistance in ABCB1-and ABCC10-overexpressing cells and tumors H Zhang, A Patel, YJ Wang, YK Zhang, RJ Kathawala, LH Qiu, BA Patel, ... Molecular cancer therapeutics 16 (6), 1021-1030, 2017 | 38 | 2017 |
| Novel 4‐thiazolidinones as non‐nucleoside inhibitors of hepatitis C virus NS5B RNA‐dependent RNA polymerase G Çakır, İ Küçükgüzel, R Guhamazumder, E Tatar, D Manvar, A Basu, ... Archiv der Pharmazie 348 (1), 10-22, 2015 | 37 | 2015 |
| The synthesis and SAR study of phenylalanine-derived (Z)-5-arylmethylidene rhodanines as anti-methicillin-resistant Staphylococcus aureus (MRSA) compounds BA Patel, CR Ashby Jr, D Hardej, TT Talele Bioorganic & medicinal chemistry letters 23 (20), 5523-5527, 2013 | 36 | 2013 |
| Design and synthesis of poly (ADP-ribose) polymerase inhibitors: impact of adenosine pocket-binding motif appendage to the 3-oxo-2, 3-dihydrobenzofuran-7-carboxamide on potency … UK Velagapudi, MF Langelier, C Delgado-Martin, ME Diolaiti, S Bakker, ... Journal of medicinal chemistry 62 (11), 5330-5357, 2019 | 34 | 2019 |
| Natural products and other inhibitors of F1FO ATP synthase BA Patel, TL D’Amico, BSJ Blagg European journal of medicinal chemistry 207, 112779, 2020 | 32 | 2020 |
| Comprehensive synthesis of amino acid-derived thiazole peptidomimetic analogues to understand the enigmatic drug/substrate-binding site of P-glycoprotein BA Patel, B Abel, AM Barbuti, UK Velagapudi, ZS Chen, SV Ambudkar, ... Journal of medicinal chemistry 61 (3), 834-864, 2018 | 27 | 2018 |
| In Vitro Antibacterial Activity of Rhodanine Derivatives against Pathogenic Clinical Isolates A AbdelKhalek, CR Ashby Jr, BA Patel, TT Talele, MN Seleem PLoS One 11 (10), e0164227, 2016 | 23 | 2016 |
| Design and synthesis of L-and D-phenylalanine derived rhodanines with novel C5-arylidenes as inhibitors of HCV NS5B polymerase BA Patel, R Krishnan, N Khadtare, KR Gurukumar, A Basu, P Arora, ... Bioorganic & medicinal chemistry 21 (11), 3262-3271, 2013 | 22 | 2013 |
| Design, Synthesis, and Biological Evaluation of (S)‐Valine Thiazole‐Derived Cyclic and Noncyclic Peptidomimetic Oligomers as Modulators of Human P … S Singh, NR Prasad, K Kapoor, EE Chufan, BA Patel, SV Ambudkar, ... ChemBioChem 15 (1), 157-169, 2014 | 21 | 2014 |
| Dual inhibition of Staphylococcus aureus DNA gyrase and topoisomerase IV activity by phenylalanine-derived (Z)-5-arylmethylidene rhodanines MM Werner, BA Patel, TT Talele, CR Ashby, Z Li, RJ Zauhar Bioorganic & Medicinal Chemistry 23 (18), 6125-6137, 2015 | 20 | 2015 |
| Thiazole-valine peptidomimetic (TTT-28) antagonizes multidrug resistance in vitro and in vivo by selectively inhibiting the efflux activity of ABCB1 YJ Wang, BA Patel, N Anreddy, YK Zhang, GN Zhang, S Alqahtani, ... Scientific reports 7 (1), 42106, 2017 | 14 | 2017 |
| Recent development in the discovery of PARP inhibitors as anticancer agents: a patent update (2016-2020) UK Velagapudi, BA Patel, X Shao, SK Pathak, DV Ferraris, TT Talele Expert Opinion on Therapeutic Patents 31 (7), 609-623, 2021 | 13 | 2021 |
| Manassantin A inhibits tumour growth under hypoxia through the activation of chaperone-mediated autophagy by modulating Hsp90 activity JK Byun, SH Lee, EJ Moon, MH Park, H Jang, DH Weitzel, HH Kim, ... British Journal of Cancer 128 (8), 1491-1502, 2023 | 3 | 2023 |
| CryoEM Structure with ATP Synthase Enables Late‐Stage Diversification of Cruentaren A X Dou, H Guo, T D'Amico, L Abdallah, C Subramanian, BA Patel, ... Chemistry–A European Journal 29 (29), e202300262, 2023 | 2 | 2023 |
| Syntheses of Enantiopure 1, 2-Ethylenediamines with Tethered Secondary Amines of the Formula H2NCH2CH [(CH2) nNHMe] NH2 (n= 1–4) from α-Amino Acids: New Agents for Asymmetric … CQ Kabes, JH Gunn, MA Selbst, RF Lucas, JA Gladysz Synthesis 52 (21), 3277-3285, 2020 | 2 | 2020 |
| Synthesis and Evaluation of Simplified Cruentaren A Analogues X Dou, BA Patel, T D’Amico, C Subramanian, E Cousineau, Y Yi, ... The Journal of Organic Chemistry 87 (15), 9940-9956, 2022 | 1 | 2022 |
| Activation of Chaperon-Mediated Autophagy Via Modulation of Hsp90 Activity Inhibits Tumor Growth Under Hypoxia JK Byun, SH Lee, EJ Moon, MH Park, H Jang, DH Weitzel, HH Kim, ... | 1 | 2021 |
